SCHEMBL9833207

SCHEMBL9833207

COc1ccc(CSc2c(C(=O)O)cccc2[N+](=O)[O-])cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.53
TSHR P16473 1/20 0.50
ALDH1A1 P00352 5/20 0.49
LMNA P02545 1/20 0.49
AKR1C3 P42330 2/20 0.46
AKR1C2 P52895 2/20 0.46
AKR1B10 O60218 1/20 0.46
AKR1B1 P15121 1/20 0.46
AKR1C4 P17516 1/20 0.46
AKR1C1 Q04828 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
PTPN1 P18031 1/20 0.44
NPC1 O15118 1/20 0.44
MAPK1 P28482 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10831867 0.89 HPGD (0.55) HPGDALDH1A1LMNASMN1; SMN2CYP3A4
SCHEMBL9087640 0.86 TSHR (0.51) HPGDTSHRALDH1A1LMNASMN1; SMN2
SCHEMBL9833015 0.82 HPGD (0.48) HPGDALDH1A1LMNASMN1; SMN2PTPN1
SCHEMBL543367 0.81 ALDH1A1 (0.54) HPGDTSHRALDH1A1LMNASMN1; SMN2
SCHEMBL30786123 0.80 TP53 (0.50) HPGDALDH1A1SMN1; SMN2USP2TP53
SCHEMBL30786121 0.80 TP53 (0.50) HPGDALDH1A1SMN1; SMN2USP2TP53
SCHEMBL31466650 0.76 HPGD (0.62) HPGDTSHRALDH1A1LMNAAKR1C3
SCHEMBL27536048 0.76 DTYMK (0.52) HPGDALDH1A1LMNAAKR1C3AKR1C2
SCHEMBL8996846 0.76 SMN1; SMN2 (0.51) HPGDALDH1A1LMNASMN1; SMN2CYP3A4
SCHEMBL7924787 0.75 TSHR (0.57) HPGDTSHRALDH1A1LMNAAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0163238-B1 SUBSTITUTED AND BRIDGED PYRIDINES USEFUL AS PHARMACEUTICAL AGENTS MERCK & CO. INC. (US) 1991-07-24 EP disclosed