SCHEMBL9833147

SCHEMBL9833147

Cc1cnc2nc(S(=O)(=O)Nc3c(C)cccc3C(=O)OCc3ccccn3)nn2c1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.36
PDE5A O76074 2/20 0.36
POLB P06746 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10666529 0.89 HPGD (0.42) PDE5APOLBLMNASMN1; SMN2NPC1
SCHEMBL9831601 0.88 LMNA (0.39) LMNASMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL10667612 0.87 PDE5A (0.36) PDE5APOLBLMNAALDH1A1TP53
SCHEMBL9831995 0.86 LMNA (0.35) PDE5APOLBLMNASMN1; SMN2NPC1
SCHEMBL9832148 0.85 FFAR4 (0.37) POLBLMNAALDH1A1MAPTKMT2A
SCHEMBL9832728 0.84 ALDH1A1 (0.48) PDE5APOLBLMNASMN1; SMN2NPC1
SCHEMBL9833209 0.84 CYP3A4 (0.37) LMNASMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL9830568 0.83 LMNA (0.36) LMNASMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL9831648 0.82 TSHR (0.48) PDE5APOLBLMNASMN1; SMN2ALDH1A1
SCHEMBL9831620 0.82 NPC1 (0.33) POLBLMNANPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed