SCHEMBL9833151

SCHEMBL9833151

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2cccc(C(F)(F)F)c2)c2c1COc1ccccc1-2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.40
MAPT P10636 5/20 0.39
POLB P06746 4/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
TP53 P04637 2/20 0.38
NPY5R Q15761 3/20 0.37
KCNJ6 P48051 2/20 0.37
KCNJ5 P48544 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833261 0.95 IDO1 (0.44) IDO1MAPTPOLBKMT2AKDM4E
SCHEMBL9831794 0.91 PTGS1 (0.42) MAPTPOLBKMT2AMEN1PTGS1
SCHEMBL9834929 0.90 CCNA2 (0.41) MAPTPOLBALDH1A1PTGS1PTGS2
SCHEMBL9316748 0.90 MAPT (0.44) MAPTPOLBKDM4EALDH1A1PTGS1
SCHEMBL9831514 0.89 MAPT (0.42) MAPTPOLBKDM4EALDH1A1TP53
SCHEMBL10568771 0.88 MAPT (0.41) MAPTPOLBSMN1; SMN2LMNATP53
SCHEMBL9833916 0.87 MAPT (0.42) MAPTPOLBKMT2AMEN1ALDH1A1
SCHEMBL9831545 0.87 RIPK1 (0.41) MAPTPOLBKDM4EALDH1A1PTGS1
SCHEMBL9832762 0.86 MAPT (0.41) MAPTPOLBKDM4EALDH1A1GLA
SCHEMBL9319611 0.86 MAPT (0.43) MAPTPOLBKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed