SCHEMBL9833283

SCHEMBL9833283

COCc1oc(-c2ccc(Cl)cc2)nc1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
LMNA P02545 2/20 0.54
KDM4E B2RXH2 6/20 0.47
TARBP2 Q15633 1/20 0.45
XBP1 P17861 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HPGD P15428 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
PPARD Q03181 3/20 0.42
PPARG P37231 3/20 0.42
PPARA Q07869 2/20 0.42
CYP2C9 P11712 1/20 0.42
KCNH2 Q12809 1/20 0.42
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
IKBKB O14920 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746500 0.85 TARBP2 (0.49) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL4427114 0.84 VDR (0.50) KDM4EPPARDPPARGPPARA
SCHEMBL9830911 0.82 KDM4E (0.50) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL18003574 0.82 ALDH1A1 (0.45) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL9831245 0.81 KDM4E (0.52) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL18003205 0.80 TARBP2 (0.44) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL9830393 0.78 ALDH1A1 (0.54) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL9833935 0.78 ALDH1A1 (0.50) ALDH1A1LMNAKDM4ETARBP2XBP1
SCHEMBL18003366 0.77 ALDH1A1 (0.56) ALDH1A1LMNAKDM4ETARBP2NPSR1
Romazarit SCHEMBL43265 0.77 ALDH1A1 (0.50) ALDH1A1LMNAKDM4ETARBP2PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed