SCHEMBL9833718

SCHEMBL9833718

O=S(=O)(NCC1CCCC(O)C1)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.51
MEN1 O00255 5/20 0.50
NPC1 O15118 1/20 0.48
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
POLB P06746 1/20 0.47
HTT P42858 2/20 0.47
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GBA1 P04062 1/20 0.47
HPGD P15428 1/20 0.46
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ALDH1A1 P00352 2/20 0.44
PKM P14618 1/20 0.44
CYP19A1 P11511 1/20 0.43
HTR1A P08908 2/20 0.43
DRD2 P14416 2/20 0.43
HTR7 P34969 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832626 0.92 CNR2 (0.53) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL6310097 0.84 CNR1 (0.48) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL6310100 0.84 KMT2A (0.53) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL6799277 0.81 GBA1 (0.69) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL9832863 0.78 THRB (0.54) KMT2AMEN1HTTLMNATSHR
SCHEMBL9833355 0.77 GBA1 (0.73) KMT2AMEN1POLBGBA1ALDH1A1
SCHEMBL9832410 0.76 CNR1 (0.48) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL14606690 0.74 GBA1 (0.59) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL9832352 0.74 CNR1 (0.55) KMT2AMEN1NPC1CNR1CNR2
SCHEMBL1594065 0.74 GBA1 (0.59) KMT2AMEN1NPC1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242518-B1 Cycloalkano[1,2-b]indole-sulfonamides BAYER AG (DE) 1991-04-10 EP disclosed
US-4988820-A Inhibiting platelet aggregation, anticoagulants, thromboxane a2 antagonist BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4965258-A Anticoagulant; thromboxane a2 antagonist BAYER AKTIENGESELLSCHAFT (DE) 1990-10-23 US disclosed
US-4904797-A REACTING A (BENZENESULFONAMIDOALKYL)CYCLOALKANO(1,2-B)INDOLE WITH ACRYLONITRILE; HYDROLYSIS, HYDROGENATION, REDUCTION BAYER AKTIENGESELLSCHAFT (DE) 1990-02-27 US disclosed
US-4827032-A INTERMEDIATES FOR ANTICOAGULANTS BAYER AKTIENGESELLSCHAFT (DE) 1989-05-02 US disclosed
EP-0242518-A1 Cycloalkano[1,2-b]indole-sulfonamides BAYER AG (DE) 1987-10-28 EP disclosed