SCHEMBL9833900

SCHEMBL9833900

CC1(C)C(=O)Nc2cc(NC(=O)c3ccccn3)c([N+](=O)[O-])cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 1/20 0.45
SNCA P37840 2/20 0.45
KDR P35968 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
HDAC1 Q13547 2/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SLC11A2 P49281 1/20 0.41
PGR P06401 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832855 0.96 AURKB (0.45) AURKBSNCAKDRKDM4EHTT
SCHEMBL9832360 0.89 AURKB (0.44) AURKBSNCAKDRKDM4EHTT
SCHEMBL10376118 0.85 HCAR3 (0.53) HTTNPC1RAB9AMAPTGAA
SCHEMBL9832573 0.84 AURKB (0.44) AURKBSNCAKDRKDM4EHTT
SCHEMBL10569985 0.84 PGR (0.39) AURKBSNCAHTTNPC1RAB9A
SCHEMBL9833023 0.83 POLB (0.43) HTTNPC1RAB9AMAPTGAA
SCHEMBL9833300 0.80 NPSR1 (0.45) KDM4EHTTMAPTGAAPGR
SCHEMBL10566877 0.79 SMN1; SMN2 (0.58) HTTNPC1RAB9AMAPTGAA
SCHEMBL9832850 0.79 POLB (0.43) HTTNPC1RAB9AMAPTGAA
SCHEMBL10566364 0.78 NPC1 (0.37) HTTNPC1RAB9AHDAC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed