SCHEMBL9834154

SCHEMBL9834154

CCC(=O)N(C)c1nc(CCl)cs1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.50
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 4/20 0.45
NPC1 O15118 6/20 0.44
RAB9A P51151 6/20 0.44
GAA P10253 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 5/20 0.38
CFTR P13569 2/20 0.38
TDP1 Q9NUW8 2/20 0.36
GFER P55789 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1860031 0.84 LMNA (0.56) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL7179302 0.76 KMT2A (0.50) LMNAKMT2AMEN1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL10957778 0.74 KMT2A (0.49) LMNAKMT2AMEN1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL7186115 0.74 KMT2A (0.49) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL10957573 0.74 RAB9A (0.41) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL21929657 0.73 LMNA (0.47) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL15689106 0.73 NPC1 (0.73) LMNAKMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL23723568 0.71 SLC12A5 (0.48) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL8627107 0.71 MEN1 (0.47) LMNAKMT2AMEN1ALDH1A1KDM4E
SCHEMBL1069018 0.71 LMNA (0.46) LMNAKMT2AMEN1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0224919-B1 NEW THIAZOLE COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-08-14 EP disclosed
US-4742057-A Antiallergic thiazole compounds FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-05-03 US disclosed
EP-0224919-A2 New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-06-10 EP disclosed