SCHEMBL9834837

SCHEMBL9834837

CC1(C)C(=O)Nc2cc3c(cc21)NC(c1ccncc1O)N3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 10/20 0.40
PDE3A Q14432 10/20 0.40
PDE4A P27815 9/20 0.40
PDE4B Q07343 9/20 0.40
PDE4C Q08493 9/20 0.40
PDE4D Q08499 9/20 0.40
ATAD2 Q6PL18 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34
PGR P06401 5/20 0.33
BMPR1B O00238 1/20 0.33
BMPR1A P36894 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
ACVR1 Q04771 1/20 0.33
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10373593 0.82 KMT2A (0.44) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832061 0.80 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
Water SCHEMBL10470996 0.79 PDE3B (0.48) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10569153 0.76 ATAD2 (0.38) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10568777 0.75 PDE3B (0.40) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832921 0.75 PDE3B (0.38) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10567876 0.75 PDE3B (0.42) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566666 0.75 ATAD2 (0.42) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10373375 0.75 KMT2A (0.47) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566029 0.74 ATAD2 (0.39) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed