SCHEMBL9832061

SCHEMBL9832061

CC1(C)C(=O)Nc2cc3c(cc21)NC(c1ccncc1)N3

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 11/20 0.49
PDE3A Q14432 11/20 0.49
PDE4A P27815 10/20 0.49
PDE4B Q07343 10/20 0.49
PDE4C Q08493 10/20 0.49
PDE4D Q08499 10/20 0.49
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ATAD2 Q6PL18 1/20 0.42
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
PGR P06401 5/20 0.38
BMPR1B O00238 1/20 0.35
BMPR1A P36894 1/20 0.35
TGFBR1 P36897 1/20 0.35
ACVRL1 P37023 1/20 0.35
ACVR1 Q04771 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL10470996 0.99 PDE3B (0.48) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9835825 0.85 PDK2 (0.50) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566029 0.85 ATAD2 (0.39) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832272 0.84 ALDH1A1 (0.41) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9833030 0.84 KDM4E (0.41) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9831453 0.83 ATAD2 (0.38) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832939 0.83 ALDH1A1 (0.43) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9829995 0.83 ALDH1A1 (0.40) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10373613 0.83 MEN1 (0.44) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10567876 0.82 PDE3B (0.42) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP claimed
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
US-4863945-A CARDIOVASCULAR DISORDERS BOEHRINGER MANNHEIM GMBH (DE) 1989-09-05 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed