SCHEMBL9836026

SCHEMBL9836026

Cc1ccc(C2=C3C(=O)N(C)C(c4ccc(C)cc4)=C3C(=O)N2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.50
HSD17B10 Q99714 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
APP P05067 1/20 0.39
F2 P00734 1/20 0.38
ELANE P08246 1/20 0.38
CTSG P08311 1/20 0.38
CMA1 P23946 1/20 0.38
CTRC Q99895 1/20 0.38
MAPT P10636 1/20 0.37
ACHE P22303 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MGLL Q99685 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12725183 0.98 PTGS2 (0.49) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL10050131 0.89 PTGS2 (0.42) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL15681729 0.89 PTGS2 (0.42) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL7067426 0.89 PTGS2 (0.42) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL12725190 0.84 PTGS2 (0.40) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL5070001 0.82 NR1H2 (0.52) PTGS2MAPTTDP1MGLLNR1H2
SCHEMBL29644702 0.81 PTGS2 (0.69) PTGS2HSD17B10CYP2D6CYP2C9HPGD
SCHEMBL14757412 0.80 EGFR (0.38) PTGS2HSD17B10HPGDMAPTTDP1
SCHEMBL16456169 0.80 SENP1 (0.45) PTGS2APPALDH1A1
SCHEMBL12725181 0.80 NR1H2 (0.50) PTGS2CTRCMAPTMGLLNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0133156-B1 1,4-DIKETOPYRROLO-(3,4-C) PYRROLES CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
US-4666455-A Compositions pigmented with N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1987-05-19 US disclosed
US-4585878-A N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1986-04-29 US disclosed