SCHEMBL9836404

SCHEMBL9836404

Nc1ncnc2c1ncn2C[C@@H]1O[C@@H]1COC(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.56
MARS1 P56192 1/20 0.54
ABCB1 P08183 1/20 0.51
GSK3A P49840 2/20 0.50
RPS6KA3 P51812 2/20 0.50
MAPK14 Q16539 2/20 0.50
ADK P55263 1/20 0.49
P2RX3 P56373 1/20 0.47
P2RX4 Q99571 1/20 0.47
P2RX2 Q9UBL9 1/20 0.47
ADORA2A P29274 1/20 0.47
PI4KA P42356 1/20 0.47
PI4K2B Q8TCG2 1/20 0.47
PI4K2A Q9BTU6 1/20 0.47
PI4KB Q9UBF8 1/20 0.47
STING1 Q86WV6 1/20 0.47
SRC P12931 1/20 0.47
KDR P35968 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836401 1.00 EGFR (0.56) EGFRMARS1ABCB1GSK3ARPS6KA3
SCHEMBL10836169 0.84 EGFR (0.56) EGFRABCB1GSK3ARPS6KA3MAPK14
SCHEMBL9837800 0.82 HDAC1 (0.46)
SCHEMBL9837796 0.82 HDAC1 (0.46)
SCHEMBL11644877 0.79 ABCB1 (0.77) ABCB1GSK3ARPS6KA3MAPK14ADORA2A
SCHEMBL441535 0.79 ABCB1 (0.77) ABCB1GSK3ARPS6KA3MAPK14ADORA2A
SCHEMBL9836909 0.78 EGFR (0.54) EGFRADORA2API4KAPI4K2BPI4K2A
SCHEMBL25101074 0.78 ABCB1 (0.60) ABCB1GSK3ARPS6KA3MAPK14P2RX3
SCHEMBL12352429 0.78 P2RX3 (0.75) ABCB1GSK3ARPS6KA3MAPK14P2RX3
SCHEMBL9189337 0.78 P2RX3 (0.75) ABCB1GSK3ARPS6KA3MAPK14P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159264-B1 ANTIVIRAL COMPOUNDS MERCK & CO. INC. (US) 1991-07-24 EP disclosed
US-4617304-A VIRICIDE; HERPES MERCK & CO., INC. (US) 1986-10-14 US disclosed
EP-0159264-A2 Antiviral compounds MERCK & CO. INC. (US) 1985-10-23 EP disclosed