SCHEMBL9836754

SCHEMBL9836754

N#CC(C(=O)Nc1ccc(F)cc1)C(=O)c1nn(-c2ccccc2)c2c1Cc1c(CO)cccc1-2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
RIPK1 Q13546 1/20 0.37
KCNJ6 P48051 2/20 0.37
KCNJ5 P48544 2/20 0.37
KCNJ3 P48549 2/20 0.37
MAPT P10636 2/20 0.36
RAB9A P51151 1/20 0.36
CNR1 P21554 1/20 0.35
P2RY1 P47900 1/20 0.35
IKBKB O14920 3/20 0.34
CCR3 P51677 1/20 0.34
PIK3CD O00329 3/20 0.34
PIK3R2 O00459 3/20 0.34
PIK3CA P42336 3/20 0.34
PIK3CB P42338 3/20 0.34
PIK3CG P48736 3/20 0.34
PIK3R5 Q8WYR1 3/20 0.34
PIK3R3 Q92569 3/20 0.34
CACNA1G O43497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9175434 0.95 PIK3CD (0.34) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9173483 0.88 IKBKB (0.38) ALDH1A1LMNARIPK1KCNJ6KCNJ5
SCHEMBL9174770 0.88 RIPK1 (0.40) ALDH1A1LMNARIPK1KCNJ6KCNJ5
SCHEMBL9173066 0.86 ALDH1A1 (0.41) ALDH1A1LMNARIPK1KCNJ6KCNJ5
SCHEMBL9171874 0.84 IKBKB (0.35) ALDH1A1LMNARIPK1RAB9AIKBKB
SCHEMBL9167849 0.84 IKBKB (0.41) ALDH1A1LMNARIPK1MAPTCNR1
SCHEMBL9167969 0.83 IKBKB (0.43) ALDH1A1LMNARIPK1KCNJ6KCNJ5
SCHEMBL9176088 0.83 IKBKB (0.39) ALDH1A1LMNARIPK1KCNJ6KCNJ5
SCHEMBL9173767 0.83 PIK3CD (0.35) ALDH1A1IKBKBPIK3CDPIK3R2PIK3CA
SCHEMBL9171740 0.83 PIK3CD (0.39) ALDH1A1RIPK1KCNJ6KCNJ5KCNJ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed