SCHEMBL9837237

SCHEMBL9837237

CCc1ccc(Nc2ccccn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51
CYP2C19 P33261 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CXCR4 P61073 1/20 0.50
MAPK10 P53779 1/20 0.50
GFER P55789 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
RAB9A P51151 3/20 0.48
GRM5 P41594 1/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPKAPK2 P49137 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12125849 0.84 RIOK2 (0.51) CYP1A2MEN1KMT2ACXCR4MAPK10
SCHEMBL5025515 0.82 MEN1 (0.50) MEN1KMT2ACXCR4MAPK10GFER
SCHEMBL154709 0.81 CXCR4 (0.49) MEN1KMT2ACXCR4MAPK10GFER
SCHEMBL904444 0.79 NPC1 (0.60) HPGDMEN1KMT2AMAPK10GFER
SCHEMBL29408382 0.79 NPC1 (0.60) HPGDMEN1KMT2AMAPK10GFER
SCHEMBL7531008 0.79 RAB9A (0.56) CYP1A2CYP3A4CYP2D6CYP2C9HPGD
SCHEMBL25201789 0.79 CXCR4 (0.56) MEN1KMT2ACXCR4MAPK10GFER
SCHEMBL14030994 0.79 MEN1 (0.43) MEN1KMT2ACXCR4MAPK10GFER
SCHEMBL31390266 0.79 MEN1 (0.59) MEN1KMT2AMAPK10GFERSMN1; SMN2
SCHEMBL29582475 0.78 MEN1 (0.64) MEN1KMT2AMAPK10GFERSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028603-A Platelet-Activating Factor Antagonist; Useful In Treatment Of Inflammatory Diseases, Allergic Diseases, Asthma, Respiratory System Disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-07-02 US disclosed
EP-0316456-A1 ESTER-SUBSTITUTED THIENOTRIAZOLODIAZEPINE COMPOUNDS AND THEIR MEDICINAL USE Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-05-24 EP disclosed