SCHEMBL9837477

SCHEMBL9837477

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2ccccc2)c2c1Cc1ccc(NC(=O)CCC(=O)O)cc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
IKBKB O14920 7/20 0.37
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R2 O00459 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3R5 Q8WYR1 1/20 0.35
PIK3R3 Q92569 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9173741 0.94 IKBKB (0.38) IKBKBNOD2NOD1PIK3CDPIK3R2
SCHEMBL9174942 0.88 IKBKB (0.38) IKBKBCYP1A2PIK3CDPIK3R2PIK3CA
SCHEMBL9524294 0.88 ADORA3 (0.34) POLBIKBKBADORA3ADORA2AADORA1
SCHEMBL9525710 0.88 MAPT (0.35) POLBIKBKBADORA3ADORA2AADORA1
SCHEMBL9174505 0.88 IKBKB (0.39) IKBKBCYP1A2ALDH1A1
SCHEMBL9173430 0.87 IKBKB (0.37) IKBKBPIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL8132620 0.87 IKBKB (0.40) IKBKBMEN1KMT2APIK3CDPIK3R2
SCHEMBL9176665 0.86 IKBKB (0.35) IKBKBMEN1KMT2APIK3CDPIK3R2
SCHEMBL9167969 0.86 IKBKB (0.43) IKBKBPIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9176690 0.86 PIK3CD (0.39) MEN1KMT2APIK3CDPIK3R2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed