SCHEMBL9837531

SCHEMBL9837531

C=Cn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC4CCC3CN4)c(F)c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
KDM4E B2RXH2 5/20 0.47
HPGD P15428 4/20 0.47
HSD17B10 Q99714 4/20 0.47
PMP22 Q01453 1/20 0.46
KCNH2 Q12809 5/20 0.45
POLB P06746 2/20 0.45
OPRM1 P35372 2/20 0.45
PRKD3 O94806 1/20 0.45
ALOX15 P16050 1/20 0.45
CLK2 P49760 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
OPRD1 P41143 1/20 0.42
TOP2A P11388 4/20 0.42
TOP2B Q02880 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378400 0.87 KCNH2 (0.56) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL9837294 0.86 KDM4E (0.64) ALDH1A1KDM4EHPGDHSD17B10PMP22
SCHEMBL9837322 0.84 KDM4E (0.60) ALDH1A1KDM4EHPGDHSD17B10PMP22
SCHEMBL9864929 0.83 KCNH2 (0.54) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL9866672 0.81 KDM4E (0.61) ALDH1A1KDM4EHPGDHSD17B10PMP22
SCHEMBL9378328 0.81 KCNH2 (0.55) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL9837602 0.78 HSD17B10 (0.64) ALDH1A1KDM4EHPGDHSD17B10PMP22
SCHEMBL9866041 0.78 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL9661855 0.78 KCNH2 (0.50) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL9838691 0.78 KDM4E (0.63) ALDH1A1KDM4EHPGDHSD17B10KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159174-B1 SUBSTITUTED NAPHTHYRIDINE-, QUINOLINE- AND BENZOXAZINE- CARBOXYLIC ACIDS AS ANTIBACTERIAL AGENTS AND PROCESSES FOR THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1991-10-23 EP disclosed
US-4571396-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1986-02-18 US disclosed
EP-0159174-A2 Substituted naphthyridine-, quinoline- and benzoxazine- carboxylic acids as antibacterial agents and processes for their production WARNER-LAMBERT COMPANY (US) 1985-10-23 EP disclosed