SCHEMBL9838696

SCHEMBL9838696

CC(=O)Nc1c(F)c(F)c(F)c2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.58
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
TOP2A P11388 3/20 0.53
TOP2B Q02880 3/20 0.53
CACNA1F O60840 1/20 0.51
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.51
CACNA1D Q01668 1/20 0.51
KCNH2 Q12809 1/20 0.51
CACNA1S Q13698 1/20 0.51
CACNA1C Q13936 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877382 0.91 GSK3B (0.53) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL7576011 0.90 GSK3B (0.66) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL9688639 0.88 GSK3B (0.60) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL9376888 0.86 GSK3B (0.53) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL7577816 0.85 ADRB2 (0.51) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL1344780 0.84 MEN1 (0.68) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL10545442 0.83 MEN1 (0.52) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL9757352 0.82 GSK3B (0.58) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL5868648 0.82 GSK3B (0.60) GSK3BMEN1KMT2ATOP2ATOP2B
SCHEMBL12674057 0.81 GSK3B (0.63) GSK3BMEN1KMT2ATOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0226961-B1 5-AMINO AND 5-HYDROXY-6,8-DIFLUOROQUINOLONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
EP-0221463-A2 Quinoline derivatives and processes for preparation thereof Dainippon Pharmaceutical Co., Ltd. (JP) 1987-05-13 EP disclosed