SCHEMBL9839846

SCHEMBL9839846

CN(C)Cc1nc(CS)cs1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.41
ACHE P22303 1/20 0.39
EPHB4 P54760 1/20 0.33
F2RL3 Q96RI0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18157890 0.86 CNR2 (0.44) CNR2ACHEEPHB4F2RL3
SCHEMBL8015431 0.81 CNR2 (0.41) CNR2ACHEEPHB4F2RL3
SCHEMBL4339516 0.81 CNR2 (0.44) CNR2ACHEEPHB4F2RL3
SCHEMBL9839838 0.81 CNR2 (0.41) CNR2ACHEEPHB4F2RL3
SCHEMBL8027980 0.81 ALDH1A1 (0.41) CNR2ACHEEPHB4
Hydrochloric Acid SCHEMBL907030 0.79 ALDH1A1 (0.43) CNR2ACHEEPHB4
Hydrochloric Acid SCHEMBL906768 0.79 ALDH1A1 (0.43) CNR2ACHEEPHB4
Hydrochloric Acid SCHEMBL8600010 0.79 CNR2 (0.43) CNR2ACHEEPHB4F2RL3
SCHEMBL19071963 0.78
SCHEMBL10426608 0.74 CNR2 (0.37) CNR2ACHEEPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0180298-B1 PYRIMIDINE COMPOUNDS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-09-25 EP disclosed
EP-0134096-B1 AMINOPYRIMIDINONE DERIVATIVES AS HISTAMINE H2-ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-02-01 EP disclosed
US-4694008-A HISTAMINE H2-ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1987-09-15 US disclosed
EP-0180298-A2 Pyrimidine compounds SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-05-07 EP disclosed