SCHEMBL9840136

SCHEMBL9840136

CC1(C)C(=O)Nc2cc(NC(=O)c3ccc(-n4ccnc4)cc3)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.49
HTT P42858 1/20 0.46
CYP3A4 P08684 1/20 0.46
BAZ2B Q9UIF8 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK2 O75116 1/20 0.45
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
MAPT P10636 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 1/20 0.43
MAPK14 Q16539 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312253 0.89 ABL1 (0.54) ROCK1KMT2AROCK2GAAMAPK14
SCHEMBL9865203 0.85 CRBN (0.47) ROCK1HTTCYP3A4BAZ2BKMT2A
SCHEMBL9840437 0.83 GAA (0.53) HTTKMT2AL3MBTL1TDP1GAA
SCHEMBL16324214 0.82 CRBN (0.56) CYP3A4BAZ2BPDE3BPDE3APDE4A
SCHEMBL9312281 0.80 NQO2 (0.51) CYP3A4KMT2AMAPK14GSK3B
SCHEMBL10477973 0.80 MEN1 (0.56) HTTCYP3A4KMT2AMAPTGAA
SCHEMBL9312304 0.78 GSK3B (0.53) HTTCYP3A4KMT2AMAPTGAA
SCHEMBL22661803 0.78 CYP3A4 (0.64) ROCK1HTTCYP3A4BAZ2BKMT2A
SCHEMBL9840703 0.77 MAPK14 (0.45) CYP3A4KMT2AMAPTMAPK14RXFP1
SCHEMBL10478082 0.77 KMT2A (0.59) CYP3A4KMT2AMAPTGAAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991001986-A1 N-(DIALKYLOXOPHOSPHINYLALKYL)-LACTAMS, PROCESS FOR PREPARING THEM AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1991-02-21 WO disclosed