SCHEMBL9840784

SCHEMBL9840784

CCCCCc1cn2c(n1)SCC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.50
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
LMNA P02545 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.47
GFER P55789 1/20 0.47
KMT2A Q03164 8/20 0.45
MEN1 O00255 7/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 3/20 0.43
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
NSD2 O96028 1/20 0.40
ALPL P05186 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13268068 0.82 MAPT (0.56) MAPTNPC1RAB9ALMNANFKB1
SCHEMBL19185513 0.74 MAPT (0.46) MAPTNPC1RAB9ALMNANFKB1
Lithium Ion SCHEMBL7175365 0.71 MAPT (0.45) MAPTNPC1RAB9ALMNANFKB1
SCHEMBL4431855 0.70 WDR5 (0.44) MAPTNPC1RAB9ALMNASMN1; SMN2
SCHEMBL8883226 0.69 LMNA (0.46) NPC1RAB9ALMNASMN1; SMN2KMT2A
SCHEMBL9747245 0.67 POLB (0.40) MAPTNPC1RAB9ALMNANFKB1
SCHEMBL9749415 0.65 MAPK14 (0.52) MAPTNPC1RAB9ALMNANFKB1
SCHEMBL8937107 0.64 KCNH2 (0.52) MAPTNPC1RAB9ALMNATP53
SCHEMBL8937080 0.64 KCNH2 (0.52) MAPTNPC1RAB9ALMNATP53
SCHEMBL18660408 0.64 TP53 (0.42) MAPTSMN1; SMN2TP53GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008390-A Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines SMITHKLINE BECKMAN CORPORATION (US) 1991-04-16 US disclosed
US-4803279-A 1.4-dihydro-4-pyridyl-substituted imidazo (2,1-b) thiazoles and the corresponding thiazines. SMITHKLINE BECKMAN CORPORATION (US) 1989-02-07 US disclosed
EP-0203787-A2 Process for preparing pyridyl-substituted imidazo[2,1-b]thiazoles and thiazines SMITHKLINE BEECHAM CORPORATION (US) 1986-12-03 EP disclosed