SCHEMBL9842686

SCHEMBL9842686

Cn1cnc2c1c(=O)n(CC1(C)OCCO1)c(=O)n2C1CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 10/20 0.43
PDE4A P27815 5/20 0.43
PDE4B Q07343 5/20 0.43
PDE4C Q08493 5/20 0.43
PDE4D Q08499 5/20 0.43
ADORA2A P29274 5/20 0.43
BLM P54132 2/20 0.43
CYP1A2 P05177 2/20 0.43
PMP22 Q01453 2/20 0.43
CYP3A4 P08684 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GLA P06280 1/20 0.39
ACHE P22303 2/20 0.39
USP2 O75604 1/20 0.39
TNF P01375 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842640 0.87 AKR1B1 (0.48) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842841 0.81 PDE4A (0.49) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842771 0.80 KMT2A (0.50) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842620 0.79 ADORA2B (0.68) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842814 0.78 PDE4A (0.58) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842817 0.76 ADORA2B (0.65) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9842796 0.75 PDE4A (0.71) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL18819579 0.72 ADORA2B (0.45) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL11174923 0.71 AKR1B1 (0.63) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL18256598 0.68 ADORA2B (0.54) ADORA2BPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0430025-A2 Xanthine compound, method for preparing thereof, and a pharmaceutical composition comprising the same HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1991-06-05 EP disclosed