SCHEMBL9842928

SCHEMBL9842928

Cc1ccc2c(-c3ccccc3C#N)scc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.38
CYP1A2 P05177 2/20 0.38
TSHR P16473 1/20 0.37
GAA P10253 3/20 0.36
KDM4E B2RXH2 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
CYP3A4 P08684 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GABRA1 P14867 3/20 0.35
GABRG2 P18507 3/20 0.35
GABRB3 P28472 3/20 0.35
GABRA2 P47869 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29038987 0.77 CYP1A2 (0.49) GRM2CYP1A2TSHRGAAKDM4E
SCHEMBL7624975 0.76 GRM2 (0.49) GRM2TSHRGAAKDM4ENPSR1
SCHEMBL9842726 0.74 TSHR (0.35) GRM2CYP1A2TSHRGAAKDM4E
SCHEMBL8550394 0.72 TSHR (0.36) GRM2CYP1A2TSHRGAAKDM4E
SCHEMBL21899538 0.72 TSHR (0.48) GRM2TSHRGAAKDM4EALDH1A1
SCHEMBL8487069 0.72 TRPA1 (0.52) CYP1A2TSHRKDM4EALDH1A1HPGD
SCHEMBL9226415 0.71 CYP1A2 (0.57) CYP1A2TSHRGAAKDM4ENPSR1
SCHEMBL8487337 0.71 CYP2A6 (0.40) TSHRGAAKDM4ENPSR1RXFP1
SCHEMBL9842740 0.70 TSHR (0.34) GRM2CYP1A2TSHRGAAKDM4E
SCHEMBL29993589 0.69 TSHR (0.50) GRM2TSHRGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0430709-A2 Benzthiophen derivatives GLAXO GROUP LIMITED (GB) 1991-06-05 EP disclosed