SCHEMBL9842935

SCHEMBL9842935

CCCC(=O)Nc1ccc(C(F)F)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.66
MAPT P10636 4/20 0.58
ALDH1A1 P00352 4/20 0.58
HPGD P15428 3/20 0.58
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
HTT P42858 2/20 0.54
THRB P10828 1/20 0.54
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28441128 0.86 MAPT (0.56) TP53MAPTALDH1A1HPGDCA12
SCHEMBL19002582 0.84 TP53 (0.68) TP53MAPTALDH1A1HPGDCA12
SCHEMBL11161614 0.81 TP53 (0.58) TP53MAPTALDH1A1HPGDCA12
SCHEMBL9429120 0.81 TSHR (0.66) MAPTALDH1A1HPGDCA1CA2
SCHEMBL8075597 0.80 TP53 (0.72) TP53MAPTALDH1A1HPGDCA12
SCHEMBL9842891 0.79 TP53 (0.60) TP53MAPTALDH1A1HPGDCA12
SCHEMBL39058 0.78 TP53 (0.75) TP53MAPTALDH1A1HPGDCA12
SCHEMBL5542468 0.78 TP53 (0.75) TP53MAPTALDH1A1HPGDCA12
SCHEMBL28675540 0.78 TP53 (0.75) TP53MAPTALDH1A1HPGDCA12
SCHEMBL8361539 0.78 TP53 (0.75) TP53MAPTALDH1A1HPGDCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed