SCHEMBL9844739

SCHEMBL9844739

CN(Cc1c[nH]c2nc(N)nc(O)c12)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 10/20 0.62
TYMS P04818 6/20 0.62
FPGS Q05932 3/20 0.59
FOLR2 P14207 2/20 0.59
FOLR1 P15328 2/20 0.59
GART P22102 2/20 0.59
ATIC P31939 2/20 0.59
SLC19A1 P41440 2/20 0.59
SLC46A1 Q96NT5 2/20 0.59
KDM4E B2RXH2 1/20 0.59
TLR4 O00206 1/20 0.59
MEN1 O00255 1/20 0.59
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
TP53 P04637 1/20 0.59
GLA P06280 1/20 0.59
POLB P06746 1/20 0.59
HMGB1 P09429 1/20 0.59
MAPT P10636 1/20 0.59
HPGD P15428 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9228615 0.89 DHFR (0.62) DHFRTYMSFPGSFOLR2FOLR1
SCHEMBL9564226 0.85 DHFR (0.73) DHFRTYMSFOLR2FOLR1GART
Pemetrexed SCHEMBL12022769 0.84 DHFR (0.83) DHFRTYMSFOLR2FOLR1GART
Pemetrexed SCHEMBL7848273 0.84 DHFR (0.83) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9042675 0.84 DHFR (0.66) DHFRTYMSFPGSFOLR2FOLR1
SCHEMBL10447943 0.83 DHFR (0.61) DHFRTYMSFOLR2FOLR1GART
SCHEMBL10447768 0.83 DHFR (0.65) DHFRTYMSFPGSFOLR2FOLR1
SCHEMBL8997255 0.82 DHFR (0.75) DHFRTYMSFOLR2FOLR1GART
SCHEMBL8997171 0.82 DHFR (0.75) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9228627 0.82 DHFR (0.54) DHFRTYMSFPGSFOLR2FOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed