SCHEMBL9844820

SCHEMBL9844820

Cn1cc(CCc2ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)cc2)c2c(O)nc(N)nc21

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.61
TYMS P04818 5/20 0.61
FOLR2 P14207 1/20 0.53
FOLR1 P15328 1/20 0.53
GART P22102 1/20 0.53
ATIC P31939 1/20 0.53
SHMT1 P34896 1/20 0.53
SLC19A1 P41440 1/20 0.53
FRK P42685 1/20 0.53
SLC46A1 Q96NT5 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844817 1.00 DHFR (0.61) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844833 0.95 DHFR (0.60) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9564175 0.92 DHFR (0.53) DHFRTYMS
SCHEMBL9844857 0.90 DHFR (0.55) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844793 0.86 DHFR (0.55) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844819 0.86 DHFR (0.51) DHFRTYMSFOLR2FOLR1GART
Butane SCHEMBL9844893 0.85 DHFR (0.55) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844850 0.85 DHFR (0.54) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844864 0.85 DHFR (0.46) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844866 0.85 DHFR (0.46) DHFRTYMSFOLR2FOLR1GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed