SCHEMBL9564175

SCHEMBL9564175

Cn1cc(Cc2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc2)c2c(O)nc(N)nc21

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 14/20 0.53
TYMS P04818 5/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844820 0.92 DHFR (0.61) DHFRTYMS
SCHEMBL9844817 0.92 DHFR (0.61) DHFRTYMS
SCHEMBL9844833 0.91 DHFR (0.60) DHFRTYMS
SCHEMBL9564148 0.84 L3MBTL1 (0.45) DHFRTYMS
SCHEMBL9564146 0.84 L3MBTL1 (0.45) DHFRTYMS
SCHEMBL9844873 0.82 DHFR (0.57) DHFRTYMS
SCHEMBL9844857 0.82 DHFR (0.55) DHFRTYMS
SCHEMBL9564226 0.81 DHFR (0.73) DHFRTYMS
SCHEMBL9844850 0.81 DHFR (0.54) DHFRTYMS
SCHEMBL9844793 0.79 DHFR (0.55) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed