SCHEMBL9844826

SCHEMBL9844826

COC(=O)c1ccc(CCCc2c[nH]c3nc(C)nc(O)c23)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.49
CYP4F2 P78329 1/20 0.49
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
CYP2C19 P33261 1/20 0.41
CKS1B P61024 1/20 0.41
SKP2 Q13309 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CCR6 P51684 1/20 0.40
HKDC1 Q2TB90 1/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8982456 0.88 CYP4A11 (0.48) CYP4A11CYP4F2ALDH1A1TP53CYP1A2
SCHEMBL9047680 0.81 DHFR (0.45) CYP1A2CYP3A4LMNADHFRTYMS
SCHEMBL14329878 0.81 DHFR (0.51) CYP4A11CYP4F2ALDH1A1TP53CYP1A2
SCHEMBL9085311 0.80 NAMPT (0.53) CYP4A11CYP4F2DHFRTYMS
SCHEMBL8982532 0.78 CYP4A11 (0.45) CYP4A11CYP4F2ALDH1A1TP53CYP1A2
SCHEMBL8982447 0.76 CYP4A11 (0.48) CYP4A11CYP4F2ALDH1A1TP53CYP1A2
SCHEMBL9045691 0.76 TYMS (0.48) DHFRTYMS
SCHEMBL9044792 0.74 TYMS (0.51) CYP1A2CYP3A4HPGDCCR6HKDC1
SCHEMBL9044536 0.73 NAMPT (0.51) CYP1A2CYP3A4LMNADHFRTYMS
SCHEMBL8855177 0.71 TYMS (0.61) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed