SCHEMBL9844834

SCHEMBL9844834

Nc1nc(N)c2c(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)csc2n1

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.69
TYMS P04818 6/20 0.61
FOLR2 P14207 1/20 0.56
FOLR1 P15328 1/20 0.56
GART P22102 1/20 0.56
ATIC P31939 1/20 0.56
SHMT1 P34896 1/20 0.56
SLC19A1 P41440 1/20 0.56
FRK P42685 1/20 0.56
SLC46A1 Q96NT5 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9227019 0.96 DHFR (0.65) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844898 0.95 DHFR (0.70) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844795 0.92 DHFR (0.60) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9226698 0.91 DHFR (0.66) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9227030 0.89 DHFR (0.56) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9227836 0.89 DHFR (0.57) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844996 0.86 DHFR (0.62) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9226710 0.84 DHFR (0.57) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9221909 0.84 DHFR (0.59) DHFRTYMSFOLR2FOLR1GART
SCHEMBL7848195 0.82 DHFR (0.84) DHFRTYMSFOLR2FOLR1GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed