SCHEMBL9844898

SCHEMBL9844898

Nc1nc(N)c2c(CCCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)csc2n1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.70
GART P22102 4/20 0.58
FOLR2 P14207 2/20 0.58
FOLR1 P15328 2/20 0.58
SLC19A1 P41440 1/20 0.57
TYMS P04818 3/20 0.56
ATIC P31939 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9226698 0.97 DHFR (0.66) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9844834 0.95 DHFR (0.69) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9844996 0.92 DHFR (0.62) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9227019 0.91 DHFR (0.65) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9226710 0.90 DHFR (0.57) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9221909 0.89 DHFR (0.59) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9844795 0.86 DHFR (0.60) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9227030 0.84 DHFR (0.56) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL9227836 0.83 DHFR (0.57) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL7835435 0.83 DHFR (0.76) DHFRGARTFOLR2FOLR1SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed