SCHEMBL9844847

SCHEMBL9844847

COC(=O)c1ccc(CC(C)c2cc3c(O)nc(N)nc3n2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.40
LNPEP Q9UIQ6 2/20 0.40
ERAP2 Q6P179 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.39
RAB9A P51151 2/20 0.38
GAA P10253 1/20 0.38
DHFR P00374 2/20 0.38
TLR8 Q9NR97 2/20 0.37
TLR7 Q9NYK1 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37
CYP2C19 P33261 1/20 0.37
CKS1B P61024 1/20 0.37
SKP2 Q13309 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844803 0.80 TP53 (0.46) TP53LNPEPLOXL2RAB9AGAA
SCHEMBL9844956 0.78 TP53 (0.41) TP53LNPEPERAP2LOXL2RAB9A
SCHEMBL9844806 0.71 NPC1 (0.39) TP53LNPEPERAP2LOXL2RAB9A
SCHEMBL9844747 0.69 CCR6 (0.45) TP53LOXL2DHFRTLR8TLR7
SCHEMBL9050614 0.68 TP53 (0.44) TP53LOXL2DHFRTLR8TLR7
SCHEMBL9844981 0.68 EGFR (0.46) TP53LOXL2RAB9AGAADHFR
SCHEMBL15502325 0.67 LCK (0.49) GAADHFRTLR8TLR7ALDH1A1
SCHEMBL9844832 0.67 TP53 (0.44) TP53LOXL2RAB9AGAADHFR
SCHEMBL9844887 0.67 CYP3A4 (0.44) TP53LOXL2RAB9AGAADHFR
SCHEMBL21667558 0.66 DHFR (0.57) TP53LOXL2GAADHFRTLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed