SCHEMBL9844747

SCHEMBL9844747

COC(=O)c1ccc(CCc2c(Br)n(C)c3nc(N)nc(O)c23)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 1/20 0.45
HKDC1 Q2TB90 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
TP53 P04637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
ALOX12 P18054 1/20 0.44
CKS1B P61024 1/20 0.44
SKP2 Q13309 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP4A11 Q02928 2/20 0.41
CYP4F2 P78329 1/20 0.41
DHFR P00374 1/20 0.40
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9556787 0.84 DRD2 (0.45) CCR6HKDC1CYP1A2CYP3A4CYP2C9
SCHEMBL9844803 0.78 TP53 (0.46) CCR6HKDC1CYP1A2CYP3A4CYP2C9
SCHEMBL14329878 0.74 DHFR (0.51) CCR6HKDC1CYP1A2CYP3A4CYP2C9
SCHEMBL8802862 0.73 TP53 (0.46) CCR6HKDC1CYP1A2CYP3A4CYP2C9
SCHEMBL9339245 0.73 CYP4A11 (0.55) CYP1A2CYP3A4CYP2C9CYP2C19TP53
SCHEMBL9339199 0.73 DHFR (0.54) CYP1A2CYP3A4CYP2C9CYP2C19TP53
SCHEMBL9844802 0.73 AGTR1 (0.40) ALDH1A1HIF1ATLR7SMN1; SMN2DRD2
SCHEMBL9341073 0.72 CYP4A11 (0.53) CYP1A2CYP3A4CYP2C9CYP2C19TP53
SCHEMBL9844887 0.69 CYP3A4 (0.44) CCR6HKDC1CYP1A2CYP3A4CYP2C9
SCHEMBL21667558 0.69 DHFR (0.57) TP53ALDH1A1DHFRTLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed