SCHEMBL9844870

SCHEMBL9844870

CN(Cc1cc2c(O)nc(N)nc2[nH]1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 7/20 0.62
SLC46A1 Q96NT5 6/20 0.59
TYMS P04818 3/20 0.59
FOLR2 P14207 2/20 0.59
SLC19A1 P41440 2/20 0.59
DHFR P00374 1/20 0.59
EHMT2 Q96KQ7 1/20 0.59
GART P22102 3/20 0.51
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844853 0.85 FOLR1 (0.62) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9844813 0.83 FOLR1 (0.68) FOLR1SLC46A1FOLR2SLC19A1GART
SCHEMBL9227335 0.78 TYMS (0.51) FOLR1SLC46A1TYMSFOLR2SLC19A1
Raltitrexed SCHEMBL12022787 0.77 TYMS (0.74) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9040482 0.77 TYMS (0.55) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9844872 0.77 TYMS (0.52) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9219313 0.76 FOLR1 (0.52) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9226749 0.76 FOLR1 (0.52) FOLR1SLC46A1TYMSFOLR2SLC19A1
SCHEMBL9844899 0.76 GART (0.68) FOLR1SLC46A1FOLR2SLC19A1GART
SCHEMBL9844849 0.76 GART (0.67) FOLR1SLC46A1TYMSFOLR2SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed