SCHEMBL9844872

SCHEMBL9844872

CN(Cc1cn(C)c2nc(N)nc(O)c12)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMS P04818 5/20 0.52
FOLR1 P15328 2/20 0.52
DHFR P00374 2/20 0.52
FOLR2 P14207 1/20 0.52
SLC19A1 P41440 1/20 0.52
EHMT2 Q96KQ7 1/20 0.52
SLC46A1 Q96NT5 1/20 0.52
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9227335 0.81 TYMS (0.51) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9564175 0.78 DHFR (0.53) TYMSDHFR
SCHEMBL9040482 0.77 TYMS (0.55) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9844817 0.77 DHFR (0.61) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9844820 0.77 DHFR (0.61) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9844870 0.77 FOLR1 (0.62) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9844873 0.77 DHFR (0.57) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9844833 0.76 DHFR (0.60) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL8325555 0.76 DHFR (0.54) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9219313 0.75 FOLR1 (0.52) TYMSFOLR1DHFRFOLR2SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed