Bromide

Bromide

SCHEMBL9845004

Br.O=C(O)c1cn(C2CC2)c2c(F)c(N3CC4=C(CNC4)C3)c(F)cc2c1=O

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.53
TOP2A P11388 7/20 0.56
TOP2B Q02880 7/20 0.56
KCNH2 Q12809 5/20 0.54
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 3/20 0.54
HPGD P15428 3/20 0.54
HSD17B10 Q99714 3/20 0.54
POLB P06746 2/20 0.54
OPRM1 P35372 2/20 0.54
PRKD3 O94806 1/20 0.54
ALOX15 P16050 1/20 0.54
CLK2 P49760 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CHRM1 P11229 1/20 0.53
OPRD1 P41143 1/20 0.53
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9693064 0.99 TOP2A (0.57) TOP2ATOP2BKCNH2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9692567 0.98 TOP2A (0.56) TOP2ATOP2BKCNH2ALDH1A1KDM4E
Formic Acid SCHEMBL9692677 0.95 TOP2A (0.53) TOP2ATOP2BKCNH2ALDH1A1KDM4E
Bromide SCHEMBL9736884 0.93 KCNH2 (0.53) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL9693045 0.92 KCNH2 (0.53) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL9690836 0.88 TOP2A (0.58) TOP2ATOP2BKCNH2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9693049 0.87 TOP2A (0.57) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL9844994 0.86 KCNH2 (0.44) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL9693034 0.85 KCNH2 (0.57) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL29638251 0.85 ALDH1A1 (0.66) TOP2ATOP2BKCNH2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0424850-A1 Quinolone compounds and a process for their preparation KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1991-05-02 EP disclosed