SCHEMBL9846214

SCHEMBL9846214

COc1nc(C)c(C(C)O)cc1C=O

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 11/20 0.35
ALDH1A1 P00352 3/20 0.33
GAA P10253 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RORC P51449 2/20 0.33
TRIM24 O15164 1/20 0.33
TYR P14679 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
PRKDC P78527 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9586039 0.77 ALDH1A1 (0.48) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL30705516 0.76 ALDH1A1 (0.39) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL9681854 0.76 ALDH1A1 (0.39) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL9267418 0.72 ALDH1A1 (0.39) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL9846110 0.72 GAA (0.55) ALDH1A1GAAKDM4E
SCHEMBL12090841 0.69 ALDH1A1 (0.39) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL30701222 0.69 ERN1 (0.46) ERN1ALDH1A1KDM4ETSHRTDP1
SCHEMBL19330163 0.69 ERN1 (0.46) ERN1ALDH1A1KDM4ETSHRTDP1
SCHEMBL9846251 0.69 GRM1 (0.37) ERN1ALDH1A1GAAKDM4ETSHR
SCHEMBL9828231 0.67 ALDH1A1 (0.55) ERN1ALDH1A1GAAKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed