SCHEMBL9846221

SCHEMBL9846221

CCCc1cc(C#N)c(Cl)nc1C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.41
KHK P50053 1/20 0.40
PGK1 P00558 1/20 0.40
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
KDM5A P29375 1/20 0.37
KDM4E B2RXH2 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23369596 0.86 POLB (0.43) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL6955377 0.86 CYP1A2 (0.51) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL9846336 0.78 GAA (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1POLB
SCHEMBL33526375 0.76 NPSR1 (0.59) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL20303775 0.74 NPSR1 (0.57) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL2394013 0.74 NPSR1 (0.57) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL30442040 0.74 NPSR1 (0.57) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL6050497 0.72 KHK (0.62) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL16370648 0.72 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL16828824 0.72 NPSR1 (0.54) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed