SCHEMBL9846226

SCHEMBL9846226

CCc1cc(C(C)c2nc3c(C)cccc3o2)c(=O)[nH]c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
PARP1 P09874 3/20 0.33
ALDH1A1 P00352 2/20 0.33
FBP1 P09467 1/20 0.33
GLA P06280 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
F2RL3 Q96RI0 1/20 0.33
ELANE P08246 4/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
PARP14 Q460N5 1/20 0.31
TNKS O95271 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30
TYMS P04818 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
HCAR2 Q8TDS4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5573692 0.84 MAPT (0.39) ALDH1A1GLAL3MBTL1ELANEKDM4E
SCHEMBL9278111 0.75 PIK3CD (0.44) PIK3CDPIK3CBPIK3CGPARP1ALDH1A1
SCHEMBL14610912 0.69 TP53 (0.42) FBP1F2RL3ELANETP53AGPAT2
SCHEMBL9846224 0.64 PARP1 (0.37) PIK3CDPIK3CBPIK3CGPARP1ALDH1A1
SCHEMBL9846133 0.64 PIK3CD (0.42) PIK3CDPIK3CBPIK3CGPARP1ALDH1A1
SCHEMBL5542360 0.63 F2RL3 (0.45) PIK3CDPIK3CBPIK3CGFBP1F2RL3
SCHEMBL9166348 0.62 IDH1 (0.37) PIK3CDPIK3CBPIK3CGPARP1ALDH1A1
SCHEMBL9166681 0.62 PIK3CD (0.41) PIK3CDPIK3CBPIK3CGPARP1ALDH1A1
SCHEMBL9442179 0.61 ELANE (0.36) ALDH1A1GLAL3MBTL1ELANEKDM4E
SCHEMBL9281338 0.61 PIK3CD (0.44) PIK3CDPIK3CBALDH1A1GLAELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed