SCHEMBL9846269

SCHEMBL9846269

COc1ccnc(OC)c1C#N

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
MAPK1 P28482 1/20 0.65
L3MBTL1 Q9Y468 1/20 0.65
KMT2A Q03164 5/20 0.63
MAPT P10636 5/20 0.63
GAA P10253 2/20 0.63
RAB9A P51151 5/20 0.60
MEN1 O00255 3/20 0.60
NPC1 O15118 2/20 0.60
HTT P42858 1/20 0.53
GFER P55789 1/20 0.49
KDM4E B2RXH2 4/20 0.48
HPGD P15428 3/20 0.48
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16121109 0.83 ALDH1A1 (0.61) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL1314187 0.82 ALDH1A1 (0.76) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL8427710 0.81 ALDH1A1 (0.58) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL676675 0.81 RECQL (0.51) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL18297669 0.81 ALDH1A1 (0.46) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL4009316 0.81 ALDH1A1 (0.74) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL16098128 0.80 RAB9A (0.55) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL441301 0.79 MAPK1 (0.51) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL768031 0.79 ALDH1A1 (0.45) ALDH1A1MAPK1L3MBTL1KMT2AMAPT
SCHEMBL31728806 0.79 ALDH1A1 (0.45) ALDH1A1MAPK1L3MBTL1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed