SCHEMBL9846629

SCHEMBL9846629

COc1ccc(CCCCOC(=O)Oc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.54
RAB9A P51151 1/20 0.54
HTR2A P28223 1/20 0.54
KCNH2 Q12809 3/20 0.52
KCNJ1 P48048 1/20 0.52
ALDH1A1 P00352 4/20 0.52
KMT2A Q03164 2/20 0.50
EPHX1 P07099 1/20 0.50
GAA P10253 2/20 0.47
MEN1 O00255 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4386673 0.91 MAPT (0.57) MAPTRAB9AHTR2AKCNH2KCNJ1
SCHEMBL14876975 0.84 HTR2A (0.54) MAPTRAB9AHTR2AALDH1A1KMT2A
SCHEMBL9223114 0.84 HTR2A (0.60) MAPTRAB9AHTR2AKCNH2KMT2A
SCHEMBL25236588 0.84 EPHX1 (0.61) KCNH2KCNJ1EPHX1
SCHEMBL10062012 0.84 HTR2A (0.56) MAPTHTR2AALDH1A1KMT2AGAA
SCHEMBL22959846 0.84 HTR2A (0.56) MAPTHTR2AALDH1A1KMT2AGAA
SCHEMBL6594172 0.83 HTR2A (0.74) MAPTRAB9AHTR2AKCNH2KCNJ1
SCHEMBL4660469 0.83 KCNH2 (0.65) MAPTRAB9AKCNH2KCNJ1ALDH1A1
SCHEMBL763025 0.83 HTR2A (0.57) MAPTHTR2AALDH1A1KMT2AGAA
SCHEMBL409598 0.83 HTR2A (0.59) MAPTHTR2AALDH1A1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429232-A1 N-substituted derivatives of 3R,4R-ethyl-[(1-methyl-1H-imidazol-5-yl)methyl]-2-pyrrolidinone ALLERGAN, INC. (US) 1991-05-29 EP disclosed