SCHEMBL9848012

SCHEMBL9848012

CCCCOC(=O)CN[C@@H](Cc1ccc(O)cc1)C(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.48
ESR2 Q92731 1/20 0.48
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47
NR1H2 P55055 1/20 0.47
RNASEL Q05823 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 2/20 0.46
KMT2A Q03164 1/20 0.46
LNPEP Q9UIQ6 3/20 0.46
MDM4 O15151 1/20 0.46
MDM2 Q00987 1/20 0.46
ERAP2 Q6P179 3/20 0.44
ERAP1 Q9NZ08 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826832 0.83 NPSR1 (0.53) ESR1ESR2CNR1CNR2TSHR
SCHEMBL8008631 0.83 NPSR1 (0.53) ESR1ESR2CNR1CNR2TSHR
SCHEMBL1721283 0.83 NPSR1 (0.53) ESR1ESR2CNR1CNR2TSHR
SCHEMBL7456029 0.82 ESR1 (0.54) ESR1ESR2CNR1CNR2TSHR
SCHEMBL7456024 0.82 ESR1 (0.54) ESR1ESR2CNR1CNR2TSHR
SCHEMBL27723176 0.80 ESR1 (0.51) ESR1ESR2CNR1CNR2TSHR
SCHEMBL7237658 0.79 ESR1 (0.59) ESR1ESR2TSHRNPSR1KMT2A
SCHEMBL8437201 0.78 IL1RN (0.50) ESR1ESR2CNR1CNR2TSHR
SCHEMBL3055258 0.76 TACR1 (0.50) ESR1ESR2CNR1CNR2TSHR
SCHEMBL3055256 0.76 TACR1 (0.50) ESR1ESR2CNR1CNR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0451422-A1 Pharmaceutically active fluoromethyltyrosine compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1991-10-16 EP disclosed