SCHEMBL9848552

SCHEMBL9848552

Nc1nnc(-c2cc(Cl)c(N)c(Cl)c2)c(N)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.53
CLK4 Q9HAZ1 1/20 0.53
CYP2D6 P10635 1/20 0.49
MAOA P21397 1/20 0.49
MAPK1 P28482 1/20 0.49
ADRA1A P35348 1/20 0.49
SCN4A P35499 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
PDE3A Q14432 1/20 0.49
SCN5A Q14524 1/20 0.49
SCN9A Q15858 1/20 0.49
SCN2A Q99250 1/20 0.49
SCN3A Q9NY46 1/20 0.49
SCN10A Q9Y5Y9 1/20 0.49
ADORA2A P29274 13/20 0.44
ADORA1 P30542 13/20 0.44
ADORA2B P29275 3/20 0.44
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929311 0.82 ADORA2A (0.62) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL6492186 0.81 CSNK1A1 (0.55) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL978678 0.79 CSNK1A1 (0.47) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL9848562 0.77 SCN9A (0.57) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL9848568 0.75 CSNK1A1 (0.41) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL9848576 0.75 CSNK1A1 (0.41) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL7349151 0.74 CSNK1A1 (0.66) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL7384520 0.74 NPC1 (0.37) ADORA2AADORA1ALDH1A1CYP3A4DHFR
SCHEMBL10843457 0.73 ADORA2A (0.71) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL12922469 0.72 CSNK1A1 (0.74) CSNK1A1CLK4CYP2D6MAOAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459829-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP claimed
EP-0459829-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed