SCHEMBL9848568

SCHEMBL9848568

CN(C)/C=N/c1c(Cl)cc(-c2nnc(N)nc2N)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
CYP2D6 P10635 1/20 0.38
MAOA P21397 1/20 0.38
MAPK1 P28482 1/20 0.38
ADRA1A P35348 1/20 0.38
SCN4A P35499 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
PDE3A Q14432 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
ADORA2A P29274 11/20 0.36
ADORA1 P30542 11/20 0.36
KMT2A Q03164 1/20 0.36
ADORA2B P29275 3/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9848576 1.00 CSNK1A1 (0.41) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL7280206 0.78 KMT2A (0.34) KMT2AKDM4EALDH1A1
SCHEMBL7280211 0.78 KMT2A (0.34) KMT2AKDM4EALDH1A1
SCHEMBL9848552 0.75 CSNK1A1 (0.53) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL7272766 0.75 ALDH1A1 (0.37) KMT2AKDM4EALDH1A1
SCHEMBL7272773 0.75 ALDH1A1 (0.37) KMT2AKDM4EALDH1A1
SCHEMBL11133814 0.73 KMT2A (0.47) MAPK1ADRA1AKMT2AKDM4EALDH1A1
SCHEMBL11133816 0.73 KMT2A (0.47) MAPK1ADRA1AKMT2AKDM4EALDH1A1
SCHEMBL3929311 0.70 ADORA2A (0.62) CSNK1A1CLK4CYP2D6MAOAMAPK1
SCHEMBL9081729 0.69 CCNA2 (0.40) MAPK1KMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459829-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed