SCHEMBL9849182

SCHEMBL9849182

N#Cc1nccc2c(O[PH](=O)O)cccc12

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.42
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
MALT1 Q9UDY8 1/20 0.34
PLAU P00749 2/20 0.33
PLCG1 P19174 1/20 0.33
ELANE P08246 4/20 0.31
AR P10275 1/20 0.31
PLAT P00750 1/20 0.30
BCAT1 P54687 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849177 0.88 CACNA2D1 (0.43) CACNA2D1KDM4EALDH1A1POLBMALT1
SCHEMBL754037 0.77 PLAU (0.50) CACNA2D1KDM4EALDH1A1POLBPLAU
SCHEMBL9849291 0.74 PLAU (0.39) KDM4EPLAUELANEPLAT
SCHEMBL7435730 0.74 KMT2A (0.56) CACNA2D1POLBELANE
SCHEMBL7438690 0.72 KDM4E (0.44) CACNA2D1KDM4EALDH1A1POLBELANE
SCHEMBL27314484 0.70 KDM4E (0.47) KDM4EALDH1A1POLBMALT1ELANE
SCHEMBL9849240 0.69 POLB (0.39) CACNA2D1KDM4EALDH1A1POLBMALT1
SCHEMBL20292623 0.68 KDM4E (0.44) CACNA2D1KDM4EALDH1A1POLBMALT1
SCHEMBL3939571 0.68 ALDH1A1 (0.48) CACNA2D1KDM4EALDH1A1POLB
SCHEMBL4856952 0.68 PLAU (0.46) CACNA2D1KDM4EALDH1A1POLBPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed