SCHEMBL9849973

SCHEMBL9849973

CN(C)C(C#N)c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
SLC6A2 P23975 6/20 0.42
SLC6A4 P31645 6/20 0.42
CHRM2 P08172 5/20 0.42
SCN1A P35498 3/20 0.42
SCN2A Q99250 3/20 0.42
SCN3A Q9NY46 3/20 0.42
KCNH2 Q12809 5/20 0.42
KCNA5 P22460 4/20 0.42
SLC6A3 Q01959 5/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2D6 P10635 3/20 0.40
KCNE1 P15382 2/20 0.40
KCNMA1 Q12791 1/20 0.38
CHRM1 P11229 4/20 0.38
HRH1 P35367 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11807865 0.82 KCNA5 (0.57) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL1998300 0.81 TSHR (0.49) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL11877693 0.76 KCNMA1 (0.35) KCNMA1
SCHEMBL702161 0.75 SMN1; SMN2 (0.49) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL22275828 0.75 SMN1; SMN2 (0.49) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL29700907 0.75 SMN1; SMN2 (0.49) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL18988389 0.74 TSHR (0.57) TSHRSLC6A2SLC6A4CHRM2SCN1A
SCHEMBL5429300 0.74 SLC6A2 (0.48) TSHRSMN1; SMN2MEN1GAAKMT2A
SCHEMBL30679621 0.74 TSHR (0.57) TSHRSLC6A2SLC6A4CHRM2SCN1A
SCHEMBL2937192 0.74 SLC6A2 (0.48) TSHRSMN1; SMN2MEN1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446097-A1 Substituted etylamines, process for their preparation, their use as therapeutic agents and intermediates for their synthesis JOUVEINAL S.A. (FR) 1991-09-11 EP disclosed
US-3956494-A ANTISECRETORY AGENTS, HETEROCYCLIC THIOPROPIONAMIDES SMITHKLINE CORPORATION (US) 1976-05-11 US disclosed
US-3950522-A N-ALKENYL OR N-ALKYNYL THIOAMIDES SMITHKLINE CORPORATION (US) 1976-04-13 US disclosed
US-3948892-A 2-Alkoxy(and 2-amino)-3-amino-2-heterocyclic-thiopropanamides SMITHKLINE CORPORATION (US) 1976-04-06 US disclosed
US-3933811-A N-aminomethyl-2-amino(and 2-amino-methyl)-2-(2-quinolyl)-thioacetamides SMITHKLINE CORPORATION (US) 1976-01-20 US disclosed