SCHEMBL9850356

SCHEMBL9850356

COc1ccc(C(N)(O)C(=O)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.54
CES2 O00748 1/20 0.54
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
PTGS2 P35354 1/20 0.49
SRC P12931 1/20 0.47
KCNK9 Q9NPC2 1/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
KIF11 P52732 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
BCHE P06276 1/20 0.45
CYP3A4 P08684 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL461653 0.82 CES1 (0.50) CES1CES2SRCCA1CA2
SCHEMBL6203510 0.82 CES1 (0.56) CES1CES2NPC1RAB9APTGS2
SCHEMBL12260648 0.80 CES1 (0.58) CES1CES2NPC1RAB9APTGS2
SCHEMBL17080312 0.80 CES1 (0.58) CES1CES2NPC1RAB9APTGS2
SCHEMBL28993094 0.79 CES1 (0.53) CES1CES2NPC1RAB9APTGS2
SCHEMBL16147101 0.79 CES1 (0.56) CES1CES2NPC1RAB9APTGS2
SCHEMBL9850344 0.78 CES1 (0.50) CES1CES2NPC1RAB9APTGS2
SCHEMBL11819939 0.74 CES1 (0.50) CES1CES2NPC1RAB9APTGS2
SCHEMBL2319756 0.73 KMT2A (0.54) CES1CES2NPC1RAB9ACDK5
SCHEMBL3939301 0.73 CES2 (0.53) CES1CES2NPC1RAB9ASRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105518001-A MODIFIED BET-PROTEIN-INHIBITING DIHYDROQUINOXALINONES AND DIHYDROPYRIDOPYRAZINONES Bayer Pharma AG 2016-04-20 CN disclosed
EP-0433112-A1 Modified gangliosides and the functional derivatives thereof FIDIA S.p.A. (IT) 1991-06-19 EP disclosed