SCHEMBL9851228

SCHEMBL9851228

COC(OC)C(CCCc1ccc(C(=O)OC(C)(C)C)cc1Cl)C(C#N)C#N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
STAT3 P40763 1/20 0.32
PDK1 Q15118 2/20 0.32
PDK2 Q15119 2/20 0.32
PDK3 Q15120 2/20 0.32
PDK4 Q16654 2/20 0.32
BUB1 O43683 1/20 0.32
SRD5A1 P18405 1/20 0.31
RAPGEF3 O95398 2/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9088289 0.82 CYP4A11 (0.41) SLC7A5CA12CA1CA2CA9
SCHEMBL9086571 0.79 CYP4A11 (0.42) SLC7A5CA12CA1CA2CA9
SCHEMBL9085713 0.78 CA12 (0.39) SLC7A5CA12CA1CA2CA9
SCHEMBL9851258 0.77 BUB1 (0.33) SLC7A5CA12CA1CA2CA9
SCHEMBL5963476 0.75 GABRA1 (0.41) SLC7A5CA12CA1CA2CA9
SCHEMBL9851250 0.74 STAT3 (0.37) SLC7A5CA12CA1CA2CA9
SCHEMBL27312730 0.73 CA12 (0.40) SLC7A5CA12CA1CA2CA9
SCHEMBL9851267 0.73 BUB1 (0.35) SLC7A5CA12CA1CA2CA9
SCHEMBL9851268 0.73 BUB1 (0.35) SLC7A5CA12CA1CA2CA9
SCHEMBL8982437 0.72 CYP4A11 (0.54) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431953-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-06-12 EP disclosed