SCHEMBL9852272

SCHEMBL9852272

Nc1nc(-c2ccc(Cl)cc2)ns1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.66
ADORA2A P29274 2/20 0.66
ADORA2B P29275 2/20 0.66
ADORA1 P30542 2/20 0.66
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP19A1 P11511 1/20 0.48
NOTUM Q6P988 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MGAM O43451 1/20 0.44
GAA P10253 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
SCN9A Q15858 1/20 0.44
ALPL P05186 1/20 0.43
LTA4H P09960 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9108544 0.80 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL11332250 0.80 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL20390644 0.80 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL20390138 0.80 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL16238754 0.80 ADORA3 (0.66) ADORA3ADORA2AADORA2BADORA1RAB9A
SCHEMBL9852130 0.79 NPC1 (0.58) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL13659745 0.79 ADORA3 (0.59) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL69810 0.79 ADORA3 (1.00) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL1219538 0.79 NPC1 (0.53) ADORA3ADORA2AADORA2BADORA1NPC1
SCHEMBL11327119 0.78 ADORA2A (0.62) ADORA3ADORA2AADORA2BADORA1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0455356-A1 Substituted 5-amino-1,2,4-thiadiazoles with pharmaceutical activity LILLY INDUSTRIES LIMITED (GB) 1991-11-06 EP disclosed
US-4259236-A COLORFAST RED SHADES ON POLYESTERS CIBA-GEIGY CORPORATION (US) 1981-03-31 US disclosed
US-4233214-A FOR POLYACRYLONITRILE AND ACID-MODIFIED POLYESTERS OR POLYAMIDES BAYER AKTIENGESELLSCHAFT (DE) 1980-11-11 US disclosed
US-4036826-A Cationic azo dyestuffs with a hydroxyalkylated ammonium group BAYER AKTIENGESELLSCHAFT (DT) 1977-07-19 US disclosed