SCHEMBL9853571

SCHEMBL9853571

c1ccc(C2CC3CCN2CC3)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.50
CHRNB2 P17787 2/20 0.50
CHRNA4 P43681 2/20 0.50
MAPT P10636 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 3/20 0.41
NPEPPS P55786 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
RIPK1 Q13546 1/20 0.38
HSD11B1 P28845 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OPRL1 P41146 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9442757 0.75 CHRNA7 (0.54) CHRNA7CHRNB2CHRNA4ALDH1A1CHRM2
Hydrochloric Acid SCHEMBL9442635 0.74 CHRNA7 (0.53) CHRNA7CHRNB2CHRNA4ALDH1A1CHRM2
SCHEMBL1217690 0.71 HRH3 (0.44) CHRNA7CHRNB2CHRNA4MAPTTDP1
SCHEMBL5228523 0.71 CHRNA7 (0.62) CHRNA7CHRNB2CHRNA4KMT2A
SCHEMBL6354340 0.70 NPEPPS (0.44) MAPTALDH1A1NPEPPSRIPK1HSD11B1
SCHEMBL6344810 0.70 CXCR4 (0.42) MAPTALDH1A1NPEPPSRIPK1HSD11B1
SCHEMBL19463939 0.70 CHRNB2 (0.56) CHRNA7CHRNB2CHRNA4MAPTTDP1
SCHEMBL12644364 0.70 CXCR4 (0.42) MAPTALDH1A1NPEPPSHSD11B1KDM4E
SCHEMBL3182932 0.70 CHRNB2 (0.56) CHRNA7CHRNB2CHRNA4MAPTTDP1
SCHEMBL14235834 0.70 CHRNB2 (0.56) CHRNA7CHRNB2CHRNA4MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0412798-A2 Substituted pyridines, their preparation, formulations and use in dementia MERCK SHARP & DOHME LTD. (GB) 1991-02-13 EP disclosed