SCHEMBL9853590

SCHEMBL9853590

Nc1cnccc1Oc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
GPBAR1 Q8TDU6 1/20 0.43
KDM4E B2RXH2 3/20 0.42
POLB P06746 1/20 0.42
HTT P42858 1/20 0.42
RAD52 P43351 1/20 0.42
KCNA3 P22001 1/20 0.41
HPGD P15428 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
KEAP1 Q14145 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9853611 0.98 CYP3A4 (0.45) CYP3A4LMNACYP1A2CYP2D6CYP2C9
SCHEMBL9853585 0.87 CYP3A4 (0.46) CYP3A4LMNACYP1A2CYP2D6CYP2C9
SCHEMBL11095020 0.81 ALDH1A1 (0.58) CYP3A4SIRT2SIRT1SIRT3KDM4E
SCHEMBL17678671 0.77 CA12 (0.39) CYP3A4LMNACYP1A2CYP2D6CYP2C9
SCHEMBL11275925 0.77 PTGS1 (0.50) CYP3A4CYP1A2CYP2C19GPBAR1HTT
SCHEMBL29577853 0.76 HTR1B (0.54) CYP3A4CYP1A2CYP2C19KDM4EKCNA3
SCHEMBL442767 0.76 HTR1B (0.54) CYP3A4CYP1A2CYP2C19KDM4EKCNA3
SCHEMBL9853600 0.75 PIN1 (0.56) LMNACYP1A2CYP2C9GPBAR1HTT
Lithium SCHEMBL6571336 0.74 HTR1B (0.52) CYP1A2CYP2C19KDM4EKCNA3HPGD
Methane SCHEMBL10959030 0.74 HTR1B (0.52) CYP1A2CYP2C19KDM4EKCNA3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4931457-A Naphthylamino-and naphthyloxy-pyridinamine comounds useful as topical antiinflammatory agents for the treatment of skin disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-05 US claimed
EP-0405426-A2 Naphthylamino- and naphthyloxy-pyridinamines and related compounds, a process for their preparation and their use as dermatological agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-02 EP disclosed
US-4931457-A Naphthylamino-and naphthyloxy-pyridinamine comounds useful as topical antiinflammatory agents for the treatment of skin disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-05 US disclosed