SCHEMBL9853716

SCHEMBL9853716

O=C(O)CNC(=O)C(CS)Nc1ncnc2[nH]cnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.39
PTGS1 P23219 1/20 0.38
GSTK1 Q9Y2Q3 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
MME P08473 4/20 0.35
ALDH1A1 P00352 3/20 0.35
ACE P12821 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.35
ECE1 P42892 1/20 0.35
BLM P54132 1/20 0.35
NPEPPS P55786 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 1/20 0.31
PTGS2 P35354 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NT5C2 P49902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9173805 0.85 SMN1; SMN2 (0.49) SMN1; SMN2ALDH1A1MAPTHPGDMAPK1
SCHEMBL9853721 0.82 SMN1; SMN2 (0.60) SMN1; SMN2MAPK1HSD17B10LMNANT5C2
SCHEMBL15730821 0.75 KDM4E (0.42) SMN1; SMN2EGLN1MAPTMAPK1HSD17B10
Glutathione SCHEMBL11157996 0.74 PTGS1 (0.66) PTGS1GSTK1EGLN1
SCHEMBL9177444 0.70 NOTUM (0.40) SMN1; SMN2EGLN1ALDH1A1HPGDMEN1
SCHEMBL19576335 0.70 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL19576298 0.70 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL19576317 0.69 SMN1; SMN2 (0.49) SMN1; SMN2HPGDHSD17B10KMT2A
SCHEMBL17234487 0.67 L3MBTL1 (0.45) EGLN1ALDH1A1MAPK1MEN1KMT2A
SCHEMBL30919984 0.67 L3MBTL1 (0.45) EGLN1ALDH1A1MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426467-A1 Prodrugs of 6-mercaptopurine and 6-thioguanine WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1991-05-08 EP disclosed