SCHEMBL9853721

SCHEMBL9853721

O=C(O)CNC(=O)[C@H](CS)Nc1ncnc2nc[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.60
BRD4 O60885 3/20 0.47
NT5C2 P49902 2/20 0.46
NT5E P21589 1/20 0.45
HSD17B10 Q99714 2/20 0.45
TSHR P16473 2/20 0.45
TP53 P04637 1/20 0.45
LMNA P02545 2/20 0.44
TOP2A P11388 2/20 0.44
BRAF P15056 2/20 0.44
CYP3A4 P08684 1/20 0.43
CYP1A2 P05177 3/20 0.42
HIF1A Q16665 1/20 0.42
CDK2 P24941 2/20 0.41
CYP2D6 P10635 1/20 0.41
MAPK1 P28482 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HTT P42858 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9853716 0.82 SMN1; SMN2 (0.39) SMN1; SMN2BRD4NT5C2HSD17B10LMNA
SCHEMBL11679062 0.76 BRD4 (0.58) SMN1; SMN2BRD4NT5C2NT5EHSD17B10
SCHEMBL30919395 0.76 TSHR (0.67) SMN1; SMN2BRD4HSD17B10TSHRTP53
SCHEMBL15709153 0.76 TSHR (0.67) SMN1; SMN2BRD4HSD17B10TSHRTP53
Glutathione SCHEMBL11158011 0.75 PTGS1 (0.65) SMN1; SMN2LMNAHDAC1HDAC2
Glutathione SCHEMBL11158003 0.75 PTGS1 (0.65) SMN1; SMN2LMNAHDAC1HDAC2
Glutathione SCHEMBL15210317 0.73 PTGS1 (0.62) SMN1; SMN2LMNA
SCHEMBL4496035 0.71 SMN1; SMN2 (0.70) SMN1; SMN2BRD4NT5C2NT5EHSD17B10
SCHEMBL9177455 0.70 HIF1A (0.57) SMN1; SMN2TSHRTP53LMNACYP1A2
SCHEMBL22118772 0.68 BRD4 (0.68) SMN1; SMN2BRD4NT5C2NT5EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426467-A1 Prodrugs of 6-mercaptopurine and 6-thioguanine WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1991-05-08 EP disclosed